SCHEMBL1645154

SCHEMBL1645154

O=C(Nc1ccccc1)c1cc(-c2cn(C3CCCCO3)nc2-c2cccc(Cl)c2)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.41
MCL1 Q07820 1/20 0.41
CNR2 P34972 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
GRM4 Q14833 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MAPK10 P53779 1/20 0.38
BRAF P15056 3/20 0.38
ACKR3 P25106 1/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
KDR P35968 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647453 0.90 CNR2 (0.41) EGFRCNR2MEN1KMT2ABRAF
SCHEMBL1646835 0.88 BRAF (0.38) EGFRCNR2BRAFATR
SCHEMBL1646072 0.88 MCL1 (0.42) MCL1MEN1KMT2APOLBGRM4
SCHEMBL1646821 0.80 MAPK14 (0.41) EGFRBRAFKDRLMNAATR
SCHEMBL1649098 0.75 ABL1 (0.41) POLBBRAF
SCHEMBL1646703 0.75 NUDT1 (0.53) BRAFCDK8KDR
SCHEMBL1938787 0.74 CNR2 (0.65) CNR2MEN1KMT2AGRM4HDAC6
SCHEMBL1645150 0.73 CSNK1D (0.40) POLBBRAFATR
SCHEMBL4291202 0.73 IRAK4 (0.40) ACKR3
SCHEMBL26112994 0.72 TP53 (0.38) ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed