SCHEMBL1646703

SCHEMBL1646703

Clc1cccc(-c2nn(C3CCCCO3)cc2-c2ccnc3[nH]ccc23)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.53
BRAF P15056 11/20 0.49
AURKB Q96GD4 3/20 0.44
AURKA O14965 2/20 0.44
CSNK1D P48730 2/20 0.42
MAPK14 Q16539 2/20 0.42
MAPK11 Q15759 1/20 0.42
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
CSF1R P07333 1/20 0.38
RET P07949 1/20 0.38
IGF1R P08069 1/20 0.38
FGFR1 P11362 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648143 0.87 BRAF (0.46) NUDT1BRAFAURKBAURKACSNK1D
SCHEMBL1647776 0.84 MAPK14 (0.59) BRAFAURKBAURKACSNK1DMAPK14
SCHEMBL1648278 0.81 AURKB (0.48) BRAFAURKBAURKACSNK1DMAPK14
SCHEMBL1646821 0.79 MAPK14 (0.41) BRAFMAPK14MAPK11KDRTP53
SCHEMBL16655108 0.77 AURKB (0.42) NUDT1BRAFAURKBAURKACSNK1D
SCHEMBL16655277 0.77 AURKB (0.44) NUDT1BRAFAURKBAURKACSNK1D
SCHEMBL1646835 0.77 BRAF (0.38) NUDT1BRAFTP53
SCHEMBL16655428 0.76 AURKB (0.46) NUDT1BRAFAURKBAURKAIKBKB
SCHEMBL1647453 0.76 CNR2 (0.41) NUDT1BRAF
SCHEMBL26112994 0.75 TP53 (0.38) MAPK14MAPK11TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2784073-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784071-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784072-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2784070-A1 3-PHENYL-4-PYRI(MI)DINYL-1H-PYRAZOLES AND THEIR USE AS FUNGICIDES Bayer CropScience AG (DE) 2014-10-01 EP disclosed
EP-2308866-A1 Phenylpyri(mi)dinylpyrazoles and their use as fungicides Bayer CropScience AG (DE) 2011-04-13 EP disclosed