SCHEMBL16474261

SCHEMBL16474261

CC(C)(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N1C[C@@H]2C[C@H]1CN2O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.44
CASP3 P42574 1/20 0.44
CASP2 P42575 1/20 0.44
CASP4 P49662 1/20 0.44
CASP5 P51878 1/20 0.44
CASP7 P55210 1/20 0.44
CASP9 P55211 1/20 0.44
CASP8 Q14790 1/20 0.44
CASP10 Q92851 1/20 0.44
CAPN1 P07384 3/20 0.43
PREP P48147 2/20 0.43
CYP3A4 P08684 4/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 2/20 0.42
TSHR P16473 2/20 0.42
POLB P06746 1/20 0.42
CYP2D6 P10635 1/20 0.42
CTSL P07711 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14964310 0.92 CASP1 (0.45) CASP1CASP3CASP2CASP4CASP5
SCHEMBL1931615 0.88 ABCB1 (0.46) CASP1CASP3CASP2CASP4CASP5
SCHEMBL7934107 0.84 CASP1 (0.44) CASP1CASP3CASP2CASP4CASP5
SCHEMBL4051763 0.82 PREP (0.43) CASP1CASP3CASP2CASP4CASP5
SCHEMBL8008130 0.82 SYK (0.45) PREPCTSL
SCHEMBL12553013 0.81 CASP1 (0.40) CASP1CASP3CASP2CASP4CASP5
SCHEMBL23386199 0.77 CASP1 (0.44) CASP1CASP3CASP2CASP4CASP5
SCHEMBL12237104 0.77 CTSL (0.47) CASP1CASP3CASP2CASP4CASP5
SCHEMBL2228500 0.76 ABCB1 (0.43) CASP1CASP3CASP2CASP4CASP5
SCHEMBL20484674 0.76 ACE (0.60) CASP1CASP3CASP2CASP4CASP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2312947-B1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2014-01-01 EP disclosed