SCHEMBL164746

SCHEMBL164746

COc1ccccc1/N=N/c1ccccc1COC(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43
NOS2 P35228 2/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
IDO1 P14902 2/20 0.41
PARP14 Q460N5 1/20 0.41
PARP10 Q53GL7 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
MAPT P10636 3/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113807 0.83 IDO1 (0.59) SMN1; SMN2LMNAKDM4ECYP1A2KMT2A
SCHEMBL22468464 0.82 KMT2A (0.48) SMN1; SMN2LMNAKDM4ECYP1A2NOS3
SCHEMBL20138424 0.82 HDAC1 (0.43) SMN1; SMN2LMNAKDM4ENOS3KMT2A
SCHEMBL22468465 0.82 KMT2A (0.48) SMN1; SMN2LMNAKDM4ECYP1A2NOS3
SCHEMBL286872 0.81 IDE (0.43) SMN1; SMN2LMNAKDM4ECYP1A2NOS3
SCHEMBL7531320 0.77 KMT2A (0.43) SMN1; SMN2LMNANOS3NOS1NOS2
SCHEMBL19973036 0.76 RXFP1 (0.48) SMN1; SMN2LMNAKDM4ECYP1A2KMT2A
SCHEMBL29501710 0.74 SMN1; SMN2 (0.48) SMN1; SMN2LMNAKDM4ECYP1A2IDO1
SCHEMBL1405477 0.74 CA1 (0.60) LMNANOS3NOS1NOS2KMT2A
SCHEMBL1405475 0.74 CA1 (0.60) LMNANOS3NOS1NOS2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 337 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024145281-A1 BIODEGRADABLE LIPIDS AND FORMULATIONS FOR INTRAMUSCULAR, IN VITRO, AND EX VIVO TRANSFECTION OF MRNA MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2024-07-04 WO disclosed
WO-2024086717-A2 HETEROARYL ENHANCERS OF THE PARTICULATE GUANYLYL CYCLASE RECEPTOR A UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2024-04-25 WO disclosed
EP-4323340-A2 E3 LIGASE BINDERS AND USES THEREOF President and Fellows of Harvard College (US) 2024-02-21 EP disclosed
WO-2023250116-A1 INDOCYANINE GREEN (ICG) MODIFICATION FOR TREATMENT OF LIVER CANCER THE CHILDREN'S MEDICAL CENTER CORPORATION (US) 2023-12-28 WO disclosed
WO-2023250342-A2 CYCLOPROPENE PHOSPHORAMIDITES AND CONJUGATES THEREOF Quantum-Si Incorporated (US) 2023-12-28 WO disclosed
EP-4288110-A2 TECHNOLOGIES FOR PREVENTING OR TREATING INFECTIONS Biohaven Therapeutics Ltd. (US) 2023-12-13 EP disclosed
EP-4248988-A2 ALKENYL SUBSTITUTED 2,5-PIPERAZINEDIONES AND THEIR USE IN COMPOSITIONS FOR DELIVERING AN AGENT TO A SUBJECT OR CELL Massachusetts Institute of Technology (US) 2023-09-27 EP disclosed
WO-2023168296-A2 CB1 LIGAND CONJUGATED COMPOUNDS AND USES THEREOF ADARX PHARMACEUTICALS, INC. (US) 2023-09-07 WO disclosed
WO-2023168045-A1 HYDROXY/AMINO OXIME-BASED HOT MELT ADHESIVES FOR REWORK, REPAIR AND RECYCLE CONAGEN INC. (US) 2023-09-07 WO disclosed
WO-2023154756-A2 THIONOLACTONES AS ADDITIVES FOR VINYL NETWORK DEGRADATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2023-08-17 WO disclosed
EP-2016044-A2 SYNTHESIS OF TETRACYCLINES AND ANALOGUES THEREOF The President and Fellows of Harvard College (US) 2009-01-21 EP disclosed
WO-2008144507-A2 SPIROOXINDOLE INHIBITORS OF AURORA KINASE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-11-27 WO disclosed
WO-2008144514-A2 POLYOL-BASED POLYMERS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2008-11-27 WO disclosed
WO-2008137692-A1 TREATMENT OF SYNUCLEINOPATHIES LINK MEDICINE CORPORATION (US) 2008-11-13 WO disclosed
WO-2008127361-A2 SYNTHESIS OF ENONE INTERMEDIATE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-10-23 WO disclosed
WO-2008122038-A1 REGULATING AUTOPHAGY PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-10-09 WO disclosed
WO-2008119015-A2 SYNTHESIS OF THIOHYDANTOINS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2008-10-02 WO disclosed
WO-2008048714-A2 BIRADICAL POLARIZING AGENTS FOR DYNAMIC NUCLEAR POLARIZATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2008-04-24 WO disclosed
WO-2007117639-A9 SYNTHESIS OF TETRACYCLINES AND ANALOGUES THEREOF HARVARD COLLEGE (US) 2008-04-17 WO disclosed
WO-2007117639-A2 SYNTHESIS OF TETRACYCLINES AND ANALOGUES THEREOF THE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2007-10-18 WO disclosed