SCHEMBL1648736

SCHEMBL1648736

COc1c(C(=O)O)ccc(CS(=O)(=O)c2ccccc2)c1-c1cnco1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 5/20 0.37
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
AAK1 Q2M2I8 2/20 0.36
ALDH1A1 P00352 3/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
EDNRA P25101 1/20 0.34
KEAP1 Q14145 4/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NFE2L2 Q16236 2/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
IMPDH1 P20839 1/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1648368 0.81 IMPDH2 (0.43) IMPDH2AAK1ROCK2ROCK1IMPDH1
SCHEMBL1649411 0.81 KMT2A (0.43) KMT2AALDH1A1L3MBTL1KEAP1NPC1
SCHEMBL1649969 0.79 KMT2A (0.35) KMT2AALDH1A1L3MBTL1KEAP1NPC1
SCHEMBL1647744 0.77 KMT2A (0.47) KMT2APOLBALDH1A1EDNRANPC1
SCHEMBL18801288 0.76 IMPDH2 (0.40) IMPDH2KMT2APOLBAAK1ROCK2
SCHEMBL1648310 0.76 KMT2A (0.35) KMT2AALDH1A1L3MBTL1KEAP1NPC1
SCHEMBL1648257 0.75 EDNRA (0.51) IMPDH2KMT2APOLBAAK1ALDH1A1
SCHEMBL1648935 0.75 KMT2A (0.41) KMT2AALDH1A1L3MBTL1KEAP1NPC1
SCHEMBL18784237 0.74 IMPDH2 (0.42) IMPDH2AAK1ROCK2ROCK1
SCHEMBL18784238 0.74 AAK1 (0.41) IMPDH2AAK1KEAP1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486004-A2 SULPHONE COMPOUNDS AND METHODS OF MAKING AND USING SAME Zafgen Corporation (US) 2012-08-15 EP disclosed
WO-2011044506-A2 SULPHONE COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN CORPORATION (US) 2011-04-14 WO disclosed