SCHEMBL16494205

SCHEMBL16494205

COCCOc1ccc2[nH]cc(CCNc3nc(N)ncc3Cc3ccc4[nH]ccc4c3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.43
CYP3A4 P08684 7/20 0.43
CYP2D6 P10635 7/20 0.43
CYP2C19 P33261 7/20 0.43
CLK4 Q9HAZ1 6/20 0.43
CYP2C9 P11712 6/20 0.43
USP2 O75604 5/20 0.43
TSHR P16473 5/20 0.43
HIF1A Q16665 5/20 0.43
MAPK1 P28482 5/20 0.43
ALDH1A1 P00352 3/20 0.43
HTR1A P08908 3/20 0.42
HTR1D P28221 3/20 0.42
HTR1B P28222 3/20 0.42
LMNA P02545 3/20 0.41
ALOX15 P16050 2/20 0.41
HTR2A P28223 3/20 0.41
HSD17B10 Q99714 4/20 0.41
IP6K1 Q92551 2/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14840209 0.92 CYP1A2 (0.51) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL16494138 0.91 CYP1A2 (0.42) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL16494349 0.89 LMNA (0.43) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL16495080 0.88 CYP1A2 (0.50) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL2598830 0.87 HTR1A (0.42) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL16494926 0.87 TRPM8 (0.51) HTR1AHTR1DHTR1BKDM4EMAPT
SCHEMBL16494750 0.86 IP6K1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL14840035 0.86 HTR2A (0.42) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL16494507 0.85 SLC6A4 (0.43) CYP1A2CYP3A4CYP2D6CYP2C19CLK4
SCHEMBL16495363 0.85 HTR1D (0.46) CYP1A2CYP3A4CYP2D6CYP2C19CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2395001-A1 Novel pyrimidine derivatives Chemilia AB (SE) 2011-12-14 EP disclosed