SCHEMBL1649446

SCHEMBL1649446

COC(=O)C1C=CN(C(=O)OC)C=C1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709284 0.77
SCHEMBL12494483 0.77 CYP2C19 (0.39) TSHRCYP2C19
SCHEMBL19346720 0.72
SCHEMBL27590444 0.70 ALDH1A1 (0.33) TSHRCYP2C19
SCHEMBL28750893 0.70 ALDH1A1 (0.33) TSHRCYP2C19
SCHEMBL12870314 0.70 ALDH1A1 (0.33) TSHRCYP2C19
SCHEMBL27608813 0.70 ALDH1A1 (0.33) TSHRCYP2C19
SCHEMBL28665742 0.69 POLB (0.42) TSHRCYP2C19
SCHEMBL9753105 0.69 TSHR (0.33) TSHR
SCHEMBL5342543 0.67 CHRNB2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
US-7790905-B2 Pharmaceutical propylene glycol solvate compositions MCNEIL-PPC, INC. (US) 2010-09-07 US disclosed