SCHEMBL16494641

SCHEMBL16494641

COc1cc(OC)c2[nH]cc(CCNc3ncc(Cc4ccc5[nH]ccc5c4)c(N)n3)c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
CSF1R P07333 2/20 0.40
NTRK2 Q16620 2/20 0.40
HTR2A P28223 5/20 0.38
HTR1A P08908 3/20 0.38
DRD2 P14416 3/20 0.38
HTR7 P34969 3/20 0.38
HTR6 P50406 3/20 0.38
DHFR P00374 1/20 0.38
HTT P42858 1/20 0.38
NTRK1 P04629 1/20 0.38
NTRK3 Q16288 1/20 0.38
USP2 O75604 5/20 0.38
CYP1A2 P05177 5/20 0.38
CYP3A4 P08684 5/20 0.38
CYP2D6 P10635 5/20 0.38
CYP2C19 P33261 5/20 0.38
CLK4 Q9HAZ1 5/20 0.38
CYP2C9 P11712 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2599419 0.92 MTNR1A (0.43) MTNR1AMTNR1BCSF1RNTRK2HTR2A
SCHEMBL2598572 0.90 HTR2A (0.44) MTNR1AMTNR1BHTR2AHTR1ADRD2
SCHEMBL14840253 0.89 HTR2A (0.50) MTNR1AMTNR1BHTR2AUSP2CYP1A2
SCHEMBL16494517 0.87 MTNR1A (0.43) MTNR1AMTNR1BCSF1RNTRK2HTR2A
SCHEMBL2598664 0.86 IP6K1 (0.47) MTNR1AMTNR1BHTR2AHTR6USP2
SCHEMBL14839743 0.83 HTR2A (0.49) MTNR1AMTNR1BHTR2AUSP2CYP1A2
SCHEMBL2598634 0.83 HTR2A (0.41) HTR2AHTR1ADHFRUSP2CYP1A2
SCHEMBL2598830 0.82 HTR1A (0.42) MTNR1AMTNR1BHTR2AHTR1AUSP2
SCHEMBL2598769 0.82 HTR2A (0.43) MTNR1AMTNR1BHTR2AHTR1ADRD2
SCHEMBL16494583 0.81 LMNA (0.43) HTR2AHTR1AUSP2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2395001-A1 Novel pyrimidine derivatives Chemilia AB (SE) 2011-12-14 EP disclosed