SCHEMBL16495384

SCHEMBL16495384

CCC(C)NC(=O)c1ccc(-c2cccc(F)c2)nc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.58
GABRA5 P31644 2/20 0.48
ROCK2 O75116 2/20 0.48
PRKG1 Q13976 2/20 0.48
PRKACA P17612 1/20 0.48
PRKACG P22612 1/20 0.48
PRKACB P22694 1/20 0.48
AKT1 P31749 1/20 0.48
DGAT1 O75907 1/20 0.48
GRM5 P41594 1/20 0.47
ALDH1A1 P00352 2/20 0.46
RAB9A P51151 1/20 0.46
BAZ2B Q9UIF8 1/20 0.46
MLNR O43193 1/20 0.45
WNT3A P56704 2/20 0.44
MAP4K4 O95819 1/20 0.44
HDAC4 P56524 1/20 0.43
CNR2 P34972 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16495932 0.88 HPGDS (0.64) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495572 0.87 GABRA5 (0.48) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495421 0.86 HPGDS (0.51) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495759 0.86 HPGDS (0.53) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495527 0.85 NPC1 (0.56) GABRA5DGAT1ALDH1A1RAB9ABAZ2B
SCHEMBL16496423 0.85 HPGDS (0.49) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495644 0.84 HPGDS (0.51) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495943 0.84 HPGDS (0.51) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495828 0.83 HPGDS (0.52) HPGDSGABRA5ROCK2PRKG1PRKACA
SCHEMBL16495568 0.83 HPGDS (0.60) HPGDSGABRA5ROCK2PRKG1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110306597-A1 Nicotinamide Derivatives CRAWFORTH JAMES MICHAEL (GB) 2011-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110306597-A1 Nicotinamide Derivatives NNT, NAMPT, NQO1 HPGDS 1073/4885GABRA5 1938/4885ROCK2 4683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.