SCHEMBL16495644

SCHEMBL16495644

CC(CCCC(C)(C)O)NC(=O)c1ccc(-c2cccc(F)c2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.51
GRM5 P41594 1/20 0.46
GABRA5 P31644 2/20 0.44
ROCK2 O75116 1/20 0.44
PRKACA P17612 1/20 0.44
PRKACG P22612 1/20 0.44
PRKACB P22694 1/20 0.44
AKT1 P31749 1/20 0.44
PRKG1 Q13976 1/20 0.44
DGAT1 O75907 1/20 0.43
MLNR O43193 1/20 0.42
WNT3A P56704 2/20 0.42
CNR2 P34972 2/20 0.42
CNR1 P21554 1/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC4 P56524 1/20 0.41
NR1I2 O75469 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16495384 0.84 HPGDS (0.58) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL16495932 0.81 HPGDS (0.64) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL16496263 0.79 HPGDS (0.55) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL16495421 0.78 HPGDS (0.51) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL16495943 0.78 HPGDS (0.51) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL2071861 0.78 HPGDS (0.66) HPGDSGABRA5PRKACGMLNRWNT3A
SCHEMBL16495693 0.77 ROCK2 (0.60) HPGDSROCK2PRKACAPRKACGPRKACB
SCHEMBL16495567 0.77 HPGDS (0.60) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL16495568 0.77 HPGDS (0.60) HPGDSGRM5GABRA5ROCK2PRKACA
SCHEMBL16496306 0.77 ADORA2A (0.49) HPGDSGRM5GABRA5ROCK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110306597-A1 Nicotinamide Derivatives CRAWFORTH JAMES MICHAEL (GB) 2011-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110306597-A1 Nicotinamide Derivatives NNT, NAMPT, NQO1 HPGDS 1073/4885GRM5 3155/4885GABRA5 1938/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.