SCHEMBL16497609

SCHEMBL16497609

C[Si](C)(C)CCOCn1c(-c2ccccc2)nc(-c2ccncc2)c1-c1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
MAPK14 Q16539 2/20 0.40
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SLC6A3 Q01959 2/20 0.39
ALOX5 P09917 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
F11 P03951 1/20 0.38
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
MAPK10 P53779 1/20 0.37
CYP17A1 P05093 1/20 0.36
LMNA P02545 2/20 0.36
HSP90AA1 P07900 1/20 0.36
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2148593 0.92 CYP1A2 (0.43) KDM4EALDH1A1HPGDMAPK14GAA
SCHEMBL16511450 0.89 MEN1 (0.36) KDM4EALDH1A1HPGDMAPK14GAA
SCHEMBL16497634 0.87 ALOX5 (0.42) KDM4EMAPK14ALOX5MEN1KMT2A
SCHEMBL14690033 0.86 DRD2 (0.38) MAPK14GAAMEN1KMT2AF11
SCHEMBL16510872 0.84 MEN1 (0.38) MAPK14MEN1KMT2AF11AKT1
SCHEMBL16497623 0.83 MEN1 (0.40) KDM4EALDH1A1HPGDMAPK14HSD17B10
SCHEMBL16511414 0.83 NPSR1 (0.40) MAPK14MEN1KMT2AF11LMNA
SCHEMBL16497631 0.83 MEN1 (0.45) MAPK14MEN1KMT2AF11AKT1
SCHEMBL16497629 0.82 BRAF (0.44) MAPK14MEN1KMT2AF11AKT1
SCHEMBL16497611 0.82 RAF1 (0.48) KDM4EALDH1A1HPGDMAPK14GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011038261-A1 HETEROCYCLIC KINASE INHIBITORS SELEXAGEN THERAPEUTICS, INC. (US) 2011-03-31 WO disclosed
WO-2011038261-A1 HETEROCYCLIC KINASE INHIBITORS SELEXAGEN THERAPEUTICS, INC. (US) 2011-03-31 WO disclosed