SCHEMBL16503576

SCHEMBL16503576

C=C(O)c1ccc2cccc(-c3c(O)cccc3Cl)c2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.35
THRB P10828 5/20 0.34
THRA P10827 4/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
WEE1 P30291 2/20 0.33
TTR P02766 2/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
CHEK1 O14757 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
GLA P06280 1/20 0.33
CYP1A2 P05177 2/20 0.33
TSHR P16473 2/20 0.33
CYP2A6 P11509 1/20 0.33
F2 P00734 1/20 0.32
PLG P00747 1/20 0.32
PLAU P00749 1/20 0.32
PLAT P00750 1/20 0.32
KLK1 P06870 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7918238 0.86 TTR (0.48) HSP90AA1THRBTHRATTRKDM4E
SCHEMBL7918472 0.83 HSD17B14 (0.36) HSP90AA1THRBCTDSP1TTRHSD17B1
SCHEMBL7918345 0.82 CYP1A2 (0.40) HSP90AA1KDM4EALDH1A1GLACYP1A2
SCHEMBL7906715 0.82 MAPT (0.41) HSP90AA1WEE1CHEK1KDM4EALDH1A1
SCHEMBL7915836 0.77 GRM2 (0.35) THRBTHRAF2PLGPLAU
SCHEMBL7917270 0.77 HTR2B (0.51)
SCHEMBL7637791 0.77 CYP1A2 (0.52) HSP90AA1THRBTHRAKDM4EALDH1A1
SCHEMBL7908665 0.77 PLA2G2D (0.49) THRBTHRATTRKDM4ETSHR
SCHEMBL16503471 0.76 DOT1L (0.39) HSP90AA1KDM4EALDH1A1TSHRF2
SCHEMBL7920129 0.74 TNF (0.45) HSD17B1HSD17B2KDM4EALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2394987-A1 ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2011-12-14 EP disclosed