SCHEMBL1650756

SCHEMBL1650756

NC(=O)N1Cc2ccccc2C=N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
SCN4A P35499 1/20 0.37
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
TRPA1 O75762 7/20 0.36
NOTUM Q6P988 2/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
PABPC1 P11940 1/20 0.33
BLM P54132 1/20 0.33
HSD17B3 P37058 2/20 0.33
NAMPT P43490 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27813867 0.86 NOTUM (0.37) TRPA1NOTUMMEN1KMT2AMAPT
SCHEMBL9387921 0.84 NOTUM (0.36) TSHRTRPA1NOTUMKDM4EALDH1A1
SCHEMBL15570101 0.83 NOTUM (0.36) LMNATSHRMAPK1SCN4ASCN5A
Hydrochloric Acid SCHEMBL28196681 0.83 NOTUM (0.35) LMNATSHRTRPA1NOTUMKDM4E
SCHEMBL27565832 0.83 NOTUM (0.47) TRPA1NOTUMHSD17B3NAMPTTAS1R3
SCHEMBL28378324 0.79 TRPA1 (0.42) LMNATRPA1NOTUMMEN1KMT2A
SCHEMBL7137593 0.79 ACHE (0.36) TSHRTRPA1NOTUMMEN1KMT2A
SCHEMBL9384425 0.79 HTR2A (0.35) TSHRTRPA1NOTUMKDM4EALDH1A1
SCHEMBL9280445 0.78 TRAP1 (0.39) LMNATSHRMAPK1MEN1KMT2A
SCHEMBL29013623 0.76 GRIN2D (0.42) LMNATSHRMAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1922183-A Nitrogenous fused heteroaromatic ring derivative BANYU PHARMA CO LTD (JP) 2007-02-28 CN claimed
US-7927613-B2 Pharmaceutical co-crystal compositions UNIVERSITY OF SOUTH FLORIDA (US) 2011-04-19 US disclosed
CN-1922183-B Nitrogenous fused heteroaromatic ring derivative BANYU PHARMA CO LTD 2010-05-26 CN disclosed
CN-1922183-A Nitrogenous fused heteroaromatic ring derivative BANYU PHARMA CO LTD (JP) 2007-02-28 CN disclosed
WO-2004069195-A2 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY DISORDERS OF THE AIRWAYS IVAX CORPORATION (US) 2004-08-19 WO disclosed