SCHEMBL16554259

SCHEMBL16554259

O=c1ccoc2cc(OCc3ccn(-c4ccccc4)n3)ccc12

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 11/20 0.52
MAOB P27338 11/20 0.52
CA12 O43570 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA5A P35218 1/20 0.47
CA7 P43166 1/20 0.47
CA5B Q9Y2D0 1/20 0.47
KDM4E B2RXH2 1/20 0.45
CA9 Q16790 1/20 0.44
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16562212 0.80 MEN1 (0.64) MAOAMAOBCA12CA1CA2
SCHEMBL29092205 0.77 MAOB (0.80) MAOAMAOBCA12CA1CA2
SCHEMBL29966607 0.77 MAOB (0.80) MAOAMAOBCA12CA1CA2
SCHEMBL10518875 0.70 DRD2 (0.63) MAOB
SCHEMBL16554123 0.70 MAOB (0.64) MAOAMAOBALDH1A1
SCHEMBL10519865 0.69 KDM4E (0.60) MAOAMAOBCA12CA1CA2
SCHEMBL10517295 0.69 DRD2 (0.67)
SCHEMBL7373528 0.68 KDM4E (0.62) MAOAMAOBCA12CA1CA2
SCHEMBL28776653 0.68 KDM4E (0.62) MAOAMAOBCA12CA1CA2
SCHEMBL17916754 0.68 GRM4 (0.46) CA12KDM4ECA9MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041470-A1 METHODS AND COMPOSITIONS FOR SELECTIVE AND TARGETED CANCER THERAPY Board Of Regents Of the University Of Texas System (US) 2016-07-13 EP disclosed
WO-2015035051-A1 METHODS AND COMPOSITIONS FOR SELECTIVE AND TARGETED CANCER THERAPY BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-03-12 WO disclosed