SCHEMBL16554398

SCHEMBL16554398

COc1ncc(N(N)C(=O)OC(C)(C)C)cc1F

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.36
PTGES2 Q9H7Z7 1/20 0.34
HDAC4 P56524 3/20 0.33
GPR52 Q9Y2T5 1/20 0.33
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
PIK3R1 P27986 2/20 0.32
MTOR P42345 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
CHRM4 P08173 1/20 0.31
S1PR3 Q99500 1/20 0.31
SYK P43405 1/20 0.31
KCNH2 Q12809 1/20 0.31
SCN5A Q14524 1/20 0.31
SCN9A Q15858 1/20 0.31
SSTR4 P31391 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14909257 0.74 PIK3CA (0.35) PIK3CAPTGES2HDAC4PIK3R1MTOR
SCHEMBL3765238 0.72 GRM2 (0.33) MTNR1AMTNR1BHDAC1HDAC8HDAC6
SCHEMBL6880953 0.71 MT-CO2 (0.36)
SCHEMBL2130967 0.71 HDAC1 (0.42) ALDH1A1HDAC1HDAC8HDAC6
SCHEMBL12140384 0.70 BRD4 (0.40) HDAC1HDAC8HDAC6
SCHEMBL14923559 0.70 SYK (0.46) PIK3CAPIK3R1MTORS1PR3SYK
SCHEMBL6879948 0.70 KIF11 (0.40) KCNH2
SCHEMBL4288276 0.70 PARP1 (0.44) MTNR1AMTNR1B
SCHEMBL30687154 0.70 SMN1; SMN2 (0.39)
SCHEMBL26939578 0.70 SMN1; SMN2 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069011-A1 NOVEL COMPOUND, METHOD FOR PREPARATION THEREOF, AND ANTIFUNGAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-05-14 WO disclosed
WO-2015034271-A1 NOVEL ANTIFUNGAL PYRIDINYLHYDRAZIDE DERIVATIVES DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2015-03-12 WO disclosed