SCHEMBL6880953

SCHEMBL6880953

CC(C)(C)OC(=O)N(N)c1ccc(Cl)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MT-CO2 P00403 1/20 0.36
PTGIR P43119 3/20 0.35
PTGDR Q13258 1/20 0.35
APP P05067 1/20 0.34
STAT3 P40763 1/20 0.33
AR P10275 2/20 0.32
TACR3 P29371 1/20 0.32
KAT6A Q92794 1/20 0.32
KAT5 Q92993 1/20 0.32
KAT8 Q9H7Z6 1/20 0.32
NR3C2 P08235 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
HTT P42858 1/20 0.31
POLB P06746 1/20 0.31
APEX1 P27695 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6881686 0.83 KDR (0.41)
SCHEMBL6879948 0.82 KIF11 (0.40) POLB
SCHEMBL2529611 0.79 MT-CO2 (0.42) MT-CO2
SCHEMBL273986 0.79 MEN1 (0.39) MT-CO2PTGIRPTGDRAPPHTT
SCHEMBL551649 0.79 MT-CO2 (0.53) MT-CO2PPARAPOLB
SCHEMBL12140384 0.77 BRD4 (0.40) MT-CO2
SCHEMBL15550751 0.77 HTR3E (0.43) MT-CO2POLB
SCHEMBL2130967 0.77 HDAC1 (0.42) PTGIRPTGDRHTT
SCHEMBL14740800 0.76 LMNA (0.34) MT-CO2POLB
SCHEMBL3765238 0.75 GRM2 (0.33) MT-CO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1474416-A1 DIHYDROBENZODIAZEPIN-2-ONE-DERIVATIVES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2004-11-10 EP disclosed
WO-2003066623-A1 DIHYDROBENZODIAZEPIN-2-ONE DERIVATIVES FOR THE TREATMENT OF NEUROLOGICAL DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2003-08-14 WO disclosed