SCHEMBL16554654

SCHEMBL16554654

COc1ccc(Cn2cc(C(N)=O)nn2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.57
MEN1 O00255 2/20 0.56
NPC1 O15118 2/20 0.56
RAB9A P51151 2/20 0.56
KMT2A Q03164 2/20 0.56
PTGS2 P35354 1/20 0.55
SNCA P37840 1/20 0.54
CA5A P35218 1/20 0.53
TUBB4A P04350 1/20 0.53
TUBB P07437 1/20 0.53
TUBA3C P0DPH7 1/20 0.53
TUBA1B P68363 1/20 0.53
TUBA4A P68366 1/20 0.53
TUBB4B P68371 1/20 0.53
TUBB3 Q13509 1/20 0.53
TUBB2A Q13885 1/20 0.53
TUBB8 Q3ZCM7 1/20 0.53
TUBA3E Q6PEY2 1/20 0.53
TUBA1A Q71U36 1/20 0.53
TUBA1C Q9BQE3 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1602886 0.87 MEN1 (0.57) MEN1NPC1RAB9AKMT2APTGS2
SCHEMBL1602867 0.87 MEN1 (0.60) MEN1NPC1RAB9AKMT2APTGS2
SCHEMBL12416497 0.86 ALDH1A1 (0.58) MEN1NPC1RAB9AKMT2APTGS2
SCHEMBL15964859 0.85 SCD (0.59) SCDMEN1NPC1RAB9AKMT2A
SCHEMBL28782136 0.84 MEN1 (0.55) MEN1NPC1RAB9AKMT2APTGS2
SCHEMBL27854173 0.84 SCD (0.61) SCDMEN1KMT2ACA5AALDH1A1
SCHEMBL13543686 0.83 HSP90AA1 (0.56) MEN1NPC1RAB9AKMT2APTGS2
SCHEMBL20344482 0.82 CA5A (0.63) SCDMEN1KMT2APTGS2CA5A
SCHEMBL1257597 0.82 ALDH1A1 (0.76) MEN1NPC1RAB9AKMT2APTGS2
SCHEMBL9857993 0.82 ALDH1A1 (0.63) SCDMEN1KMT2APTGS2CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041843-A1 NOVEL TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2016-07-13 EP disclosed
WO-2015032769-A1 NOVEL TRIAZOLO[4,5-D]PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2015-03-12 WO disclosed