SCHEMBL28782136

SCHEMBL28782136

CCC(=O)c1cn(Cc2ccc(OC)cc2)nn1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.53
SNCA P37840 1/20 0.53
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52
TUBB3 Q13509 1/20 0.52
TUBB2A Q13885 1/20 0.52
TUBB8 Q3ZCM7 1/20 0.52
TUBA3E Q6PEY2 1/20 0.52
TUBA1A Q71U36 1/20 0.52
TUBA1C Q9BQE3 1/20 0.52
TUBB6 Q9BUF5 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1602886 0.86 MEN1 (0.57) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL1602867 0.86 MEN1 (0.60) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL16554654 0.84 SCD (0.57) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL12416497 0.84 ALDH1A1 (0.58) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL24310716 0.84 ALDH1A1 (0.68) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL1257597 0.84 ALDH1A1 (0.76) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL13543686 0.82 HSP90AA1 (0.56) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL1602722 0.80 MEN1 (0.52) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL1602861 0.80 MARK4 (0.49) MEN1KMT2ANPC1RAB9AALDH1A1
SCHEMBL2511099 0.77 L3MBTL1 (0.56) MEN1KMT2ANPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101511812-A Pyrazole derivatives as cytochrome P450 inhibitors PFIZER PROD INC (US) 2009-08-19 CN disclosed