SCHEMBL16573306

SCHEMBL16573306

CNC(=O)CCc1ccc(NC(C)=S)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.51
HDAC6 Q9UBN7 5/20 0.51
HDAC3 O15379 4/20 0.51
HDAC4 P56524 4/20 0.51
HDAC7 Q8WUI4 4/20 0.51
HDAC2 Q92769 4/20 0.51
HDAC10 Q969S8 4/20 0.51
HDAC11 Q96DB2 4/20 0.51
HDAC8 Q9BY41 4/20 0.51
HDAC9 Q9UKV0 4/20 0.51
HDAC5 Q9UQL6 4/20 0.51
POLB P06746 3/20 0.50
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
RAB9A P51151 1/20 0.46
FFAR1 O14842 1/20 0.45
CYP2C9 P11712 1/20 0.45
GAA P10253 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
TAS2R38 P59533 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14387746 0.82 HDAC1 (0.53) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL16573285 0.82 ALDH1A1 (0.48) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL16573271 0.77 POLB (0.49) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL12507197 0.75 POLB (0.59) HDAC1POLBMAPTFFAR1GAA
SCHEMBL13609517 0.75 HDAC2 (0.62) HDAC1HDAC2HDAC8POLBMAPT
SCHEMBL16573272 0.75 EPHX2 (0.55) POLBMAPTHTT
SCHEMBL12237102 0.75 POLB (0.54) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL8031664 0.74 ALDH1A1 (0.43) POLBMAPTRAB9ATAS2R38
SCHEMBL12228279 0.74 HPGD (0.56) FFAR1GAA
SCHEMBL1128782 0.74 TAAR1 (0.52) HDAC1HDAC6HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2444085-B1 Diarylhydantoin compounds as androgen receptor antagonists for treatment of cancer UNIV CALIFORNIA (US) 2015-03-18 EP disclosed