SCHEMBL16584875

SCHEMBL16584875

Cc1cccc2nc(CCCNC(=O)O)n(C3CC3)c(=O)c12

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.41
PIK3CD O00329 7/20 0.41
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 2/20 0.39
HTR1A P08908 1/20 0.38
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
CASR P41180 1/20 0.38
TRPA1 O75762 1/20 0.37
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18076637 0.94 PIK3CD (0.42) PIK3CDTP53CASRTRPA1MAPT
SCHEMBL16584901 0.88 ALDH1A1 (0.39) PIK3CDLMNATSHRNPSR1MTNR1A
SCHEMBL16584903 0.88 ALDH1A1 (0.39) PIK3CDLMNATSHRNPSR1MTNR1A
SCHEMBL21178492 0.86 NPSR1 (0.38) SMN1; SMN2PIK3CDLMNATSHRNPSR1
SCHEMBL18076647 0.84 TSHR (0.51) SMN1; SMN2LMNATSHRNPSR1POLB
SCHEMBL21178494 0.83 PIK3CD (0.44) PIK3CDLMNATSHRNPSR1TP53
SCHEMBL16597161 0.82 ALDH1A1 (0.48) SMN1; SMN2PIK3CDLMNANPSR1HTR1A
SCHEMBL18076641 0.82 PIK3CD (0.39) PIK3CDTP53MAPTPOLBHRH3
SCHEMBL16584926 0.82 PIK3CD (0.40) PIK3CDTP53POLBHRH3
SCHEMBL16584911 0.81 PIK3CD (0.42) SMN1; SMN2PIK3CDLMNANPSR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3046563-A1 SUBSTITUTED AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE Calitor Sciences, LLC (US) 2016-07-27 EP disclosed
WO-2015042077-A1 SUBSTITUTED AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE CALITOR SCIENCES, LLC (US) 2015-03-26 WO disclosed