SCHEMBL16585641

SCHEMBL16585641

Cc1cnc(Cl)nc1-c1ccc(CNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 16/20 0.51
L3MBTL1 Q9Y468 1/20 0.47
STK17B O94768 1/20 0.47
STK17A Q9UEE5 1/20 0.47
PDK2 Q15119 2/20 0.46
PDK3 Q15120 2/20 0.46
PDK4 Q16654 2/20 0.46
GAA P10253 1/20 0.45
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16585497 0.94 PDK1 (0.47) PDK1L3MBTL1STK17BSTK17APDK2
SCHEMBL31380404 0.90 STK17B (0.53) PDK1L3MBTL1STK17BSTK17AGAA
SCHEMBL16793957 0.86 STK17B (0.44) PDK1STK17BSTK17APDK2PDK3
SCHEMBL16586284 0.82 MAPKAPK2 (0.47) STK17BSTK17ANAMPT
SCHEMBL12921676 0.79 AAK1 (0.53) L3MBTL1STK17BSTK17AGAANAMPT
SCHEMBL1585183 0.77 STK17B (0.52) L3MBTL1STK17BSTK17AGAANAMPT
SCHEMBL16038520 0.77 GAA (0.52) L3MBTL1GAANAMPT
SCHEMBL16794337 0.77 TRPV1 (0.42) STK17BSTK17A
SCHEMBL3180689 0.75 L3MBTL1 (0.61) L3MBTL1GAANAMPT
SCHEMBL506742 0.75 L3MBTL1 (0.53) L3MBTL1STK17BSTK17AGAANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015040425-A1 RESORCINOL N-ARYL AMIDE COMPOUNDS, FOR USE AS PYRUVATE DEHYDROGENASE KINASE INHIBITORS VERNALIS (R&D) LIMITED (GB) 2015-03-26 WO disclosed