SCHEMBL16586992

SCHEMBL16586992

CC(C)(C)OC(=O)NC(CCN1C(=O)CCC1=O)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.42
PPARA Q07869 7/20 0.42
PPARG P37231 6/20 0.42
IDO1 P14902 1/20 0.41
CTSS P25774 5/20 0.41
CTSK P43235 5/20 0.41
ACE P12821 1/20 0.41
SCN9A Q15858 1/20 0.41
ITGA4 P13612 1/20 0.41
ITGB7 P26010 1/20 0.41
PPARD Q03181 2/20 0.40
ITGAV P06756 1/20 0.39
ITGB6 P18564 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5262244 0.86 PPARA (0.43) AKT1PPARAPPARGIDO1CTSS
SCHEMBL28255277 0.86 ITGB3 (0.41) AKT1PPARAPPARGIDO1CTSK
SCHEMBL10077573 0.84 AKT1 (0.58) AKT1PPARAPPARGIDO1CTSS
SCHEMBL31004971 0.84 AKT1 (0.58) AKT1PPARAPPARGIDO1CTSS
SCHEMBL10350890 0.82 CTSK (0.51) PPARAPPARGIDO1CTSSCTSK
SCHEMBL8869903 0.82 CTSK (0.51) PPARAPPARGIDO1CTSSCTSK
SCHEMBL1262439 0.81 CTSS (0.41) PPARAPPARGIDO1CTSSCTSK
SCHEMBL5973148 0.81 FOLH1 (0.43) PPARAPPARGIDO1CTSSCTSK
SCHEMBL29695475 0.80 PPARA (0.41) PPARAPPARGIDO1CTSSCTSK
SCHEMBL31649054 0.80 AKT1 (0.49) AKT1PPARAPPARGIDO1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3046563-A1 SUBSTITUTED AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE Calitor Sciences, LLC (US) 2016-07-27 EP disclosed
WO-2015042077-A1 SUBSTITUTED AMINOPYRIMIDINE COMPOUNDS AND METHODS OF USE CALITOR SCIENCES, LLC (US) 2015-03-26 WO disclosed