SCHEMBL1658941

SCHEMBL1658941

CS(=O)(=O)Nc1c(F)cc(CCNC(=O)c2coc(Oc3cccc(Cl)c3)n2)cc1F

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 2/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
MAPT P10636 1/20 0.37
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
NPC1 O15118 1/20 0.37
THRB P10828 1/20 0.37
RAB9A P51151 1/20 0.37
POLB P06746 1/20 0.37
TRPV1 Q8NER1 3/20 0.36
HIF1A Q16665 1/20 0.36
SCN9A Q15858 2/20 0.36
TBXA2R P21731 1/20 0.35
LMNA P02545 2/20 0.35
TP53 P04637 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1659194 0.90 KLKB1 (0.40) KLKB1MAPTALDH1A1SMN1; SMN2NPC1
SCHEMBL1659330 0.90 POLB (0.40) KLKB1SMN1; SMN2NPC1RAB9APOLB
SCHEMBL1659509 0.89 KLKB1 (0.39) KLKB1POLB
SCHEMBL1661398 0.89 KLKB1 (0.39) KLKB1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL1660515 0.88 SCN9A (0.40) KLKB1RAB9APOLBSCN9A
SCHEMBL1660390 0.87 KLKB1 (0.38) KLKB1POLBTRPV1SCN9A
SCHEMBL1661096 0.86 KLKB1 (0.37) KLKB1POLBTRPV1SCN9ATBXA2R
SCHEMBL1659442 0.86 KLKB1 (0.37) KLKB1POLBTRPV1SCN9A
SCHEMBL1662387 0.84 SCN9A (0.39) KLKB1MAPTALDH1A1SMN1; SMN2NPC1
SCHEMBL1660378 0.84 MAPT (0.45) MAPTALDH1A1SMN1; SMN2NPC1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307394-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2011-04-13 EP disclosed