SCHEMBL1659442

SCHEMBL1659442

CS(=O)(=O)Nc1c(F)cc(CCNC(=O)c2coc(Oc3cccc(C4CCC4)c3)n2)cc1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.37
POLB P06746 1/20 0.34
GSK3B P49841 2/20 0.34
NLRP3 Q96P20 1/20 0.34
SCN9A Q15858 2/20 0.33
TRPV1 Q8NER1 2/20 0.32
SLC8A1 P32418 3/20 0.32
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
HCRTR2 O43614 1/20 0.31
DHODH Q02127 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661096 0.98 KLKB1 (0.37) KLKB1POLBGSK3BNLRP3SCN9A
SCHEMBL1660390 0.97 KLKB1 (0.38) KLKB1POLBGSK3BSCN9ATRPV1
SCHEMBL1659330 0.86 POLB (0.40) KLKB1POLBSCN9ACA1CA2
SCHEMBL1658941 0.86 KLKB1 (0.40) KLKB1POLBSCN9ATRPV1
SCHEMBL1659194 0.86 KLKB1 (0.40) KLKB1POLBSCN9ACA1CA2
SCHEMBL1661398 0.84 KLKB1 (0.39) KLKB1POLBSCN9ATRPV1CA1
SCHEMBL1659509 0.84 KLKB1 (0.39) KLKB1POLB
SCHEMBL12604728 0.84 PDE2A (0.37) KLKB1NLRP3
SCHEMBL1986987 0.84 PDE2A (0.37) KLKB1NLRP3
SCHEMBL1660515 0.84 SCN9A (0.40) KLKB1POLBSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307394-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2011-04-13 EP disclosed