SCHEMBL1661398

SCHEMBL1661398

CC(C)c1cccc(Oc2nc(C(=O)NCCc3cc(F)c(NS(C)(=O)=O)c(F)c3)co2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.39
POLB P06746 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GLI1 P08151 1/20 0.35
GLI2 P10070 1/20 0.35
SCN9A Q15858 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
ADORA2B P29275 1/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1988531 0.92 KLKB1 (0.43) KLKB1POLBTRPV1ADORA2BSMN1; SMN2
SCHEMBL1659330 0.89 POLB (0.40) KLKB1POLBNPC1RAB9ASCN9A
SCHEMBL1659194 0.89 KLKB1 (0.40) KLKB1POLBNPC1RAB9ASCN9A
SCHEMBL1658941 0.89 KLKB1 (0.40) KLKB1POLBNPC1RAB9ASCN9A
SCHEMBL1659509 0.87 KLKB1 (0.39) KLKB1POLB
SCHEMBL1660515 0.86 SCN9A (0.40) KLKB1POLBRAB9ASCN9AADORA2B
SCHEMBL1660390 0.86 KLKB1 (0.38) KLKB1POLBSCN9ATRPV1CA1
SCHEMBL1986290 0.85 KCNQ3 (0.41) KLKB1CA2MAPK1
SCHEMBL12603590 0.85 KCNQ3 (0.41) KLKB1CA2MAPK1
SCHEMBL1660628 0.85 CES2 (0.40) KLKB1POLBNPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307394-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2011-04-13 EP disclosed