SCHEMBL1659330

SCHEMBL1659330

CCc1cccc(Oc2nc(C(=O)NCCc3cc(F)c(NS(C)(=O)=O)c(F)c3)co2)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
KLKB1 P03952 1/20 0.40
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA7 P43166 3/20 0.38
CA9 Q16790 3/20 0.38
CA14 Q9ULX7 3/20 0.38
SCN9A Q15858 2/20 0.35
NR3C1 P04150 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NAMPT P43490 1/20 0.34
BCHE P06276 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1659194 0.90 KLKB1 (0.40) POLBKLKB1CA1CA2CA7
SCHEMBL1658941 0.90 KLKB1 (0.40) POLBKLKB1SCN9ANPC1RAB9A
SCHEMBL1659509 0.89 KLKB1 (0.39) POLBKLKB1
SCHEMBL1661398 0.89 KLKB1 (0.39) POLBKLKB1CA1CA2CA7
SCHEMBL1660515 0.88 SCN9A (0.40) POLBKLKB1SCN9ARAB9A
SCHEMBL1660390 0.87 KLKB1 (0.38) POLBKLKB1CA1CA2CA7
SCHEMBL1659442 0.86 KLKB1 (0.37) POLBKLKB1CA1CA2CA7
SCHEMBL1661096 0.86 KLKB1 (0.37) POLBKLKB1CA1CA2CA7
SCHEMBL12697436 0.84 KCNQ3 (0.38) KLKB1
SCHEMBL1985034 0.84 KCNQ3 (0.38) KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307394-A2 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2011-04-13 EP disclosed