SCHEMBL16592103

SCHEMBL16592103

NCCOc1ncc(C(F)(F)F)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C19 P33261 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.50
MRGPRX4 Q96LA9 1/20 0.48
RAB9A P51151 1/20 0.48
ALDH1A1 P00352 3/20 0.47
HPGD P15428 2/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
PLAU P00749 1/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
LMNA P02545 2/20 0.44
HTT P42858 2/20 0.43
GAA P10253 1/20 0.43
SCN9A Q15858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22809511 0.92 CYP1A2 (0.51) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
SCHEMBL22809483 0.89 CYP1A2 (0.42) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
SCHEMBL19664461 0.84 SMN1; SMN2 (0.53) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
SCHEMBL13197550 0.84 CYP1A2 (0.52) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
SCHEMBL22809399 0.83 CYP1A2 (0.38) CYP1A2CYP3A4CYP2C19SMN1; SMN2RAB9A
SCHEMBL29025473 0.83 SMN1; SMN2 (0.52) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
SCHEMBL30433202 0.83 SMN1; SMN2 (0.52) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
SCHEMBL16592086 0.83 SMN1; SMN2 (0.52) CYP1A2CYP3A4CYP2C19SMN1; SMN2MRGPRX4
Hydrochloric Acid SCHEMBL28354555 0.82 IDO1 (0.38) CYP1A2CYP3A4CYP2C19SMN1; SMN2RAB9A
Hydrochloric Acid SCHEMBL30449797 0.82 IDO1 (0.38) CYP1A2CYP3A4CYP2C19SMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776427-B Pyrimidine diamine compound and application thereof 沈阳中化农药化工研发有限公司 2022-08-23 CN disclosed
US-11154544-B2 Amide derivatives as Nav1.7 and Nav1.8 blockers RAQUALIA PHARMA INC. (JP) 2021-10-26 US disclosed
EP-3487839-B1 AMIDE DERIVATIVES AS NAV1.7 AND NAV1.8 BLOCKERS RAQUALIA PHARMA INC (JP) 2020-12-23 EP disclosed
US-9332754-B2 Alkyl phenyl sulfide derivative and pest control agent KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 2016-05-10 US disclosed
US-20150087833-A1 ALKYL PHENYL SULFIDE DERIVATIVE AND PEST CONTROL AGENT IHARA CHEMICAL INDUSTRY CO., LTD. (JP) 2015-03-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11154544-B2 Amide derivatives as Nav1.7 and Nav1.8 blockers SCN8A, SCN7A, SCN1A CYP1A2 2057/4885CYP3A4 2509/4885CYP2C19 3638/4885
US-20150087833-A1 ALKYL PHENYL SULFIDE DERIVATIVE AND PEST CONTROL AGENT C1S, TRPA1, STK39 CYP1A2 1244/4885CYP3A4 1870/4885CYP2C19 1332/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.