SCHEMBL16596178

SCHEMBL16596178

Oc1cccc(-n2nnc3ccccc32)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NT5E P21589 4/20 0.58
KCNMA1 Q12791 1/20 0.54
FGFR1 P11362 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.50
KDM4E B2RXH2 1/20 0.47
NPC1 O15118 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
RAB9A P51151 1/20 0.46
POLB P06746 1/20 0.46
MAPK1 P28482 1/20 0.46
ATM Q13315 1/20 0.46
SLC9A1 P19634 1/20 0.46
KEAP1 Q14145 1/20 0.46
ALDH1A1 P00352 3/20 0.45
TSHR P16473 1/20 0.43
DGAT1 O75907 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13338045 0.83 KCNMA1 (0.50) NT5EKCNMA1FGFR1SMN1; SMN2KDM4E
SCHEMBL503004 0.81 KCNMA1 (0.59) KCNMA1FGFR1SMN1; SMN2KDM4ENPC1
SCHEMBL18494383 0.81 KCNMA1 (0.51) NT5EKCNMA1FGFR1SMN1; SMN2KDM4E
SCHEMBL28099573 0.80 IDO1 (0.55) NT5EKCNMA1FGFR1SMN1; SMN2KDM4E
SCHEMBL241393 0.80 IDO1 (0.54) KCNMA1SMN1; SMN2KDM4ENPC1L3MBTL1
SCHEMBL2627246 0.80 KDM4E (0.64) KCNMA1SMN1; SMN2KDM4ENPC1L3MBTL1
SCHEMBL12204569 0.80 RAB9A (0.56) KCNMA1SMN1; SMN2KDM4ENPC1L3MBTL1
SCHEMBL165333 0.80 SMN1; SMN2 (0.71) KCNMA1SMN1; SMN2KDM4ENPC1L3MBTL1
SCHEMBL13191549 0.80 KCNMA1 (0.54) NT5EKCNMA1SMN1; SMN2KDM4ENPC1
SCHEMBL12204565 0.78 SMN1; SMN2 (0.62) KCNMA1SMN1; SMN2KDM4ENPC1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015042363-A1 MOLECULES AND COMPOSITIONS THAT INHIBIT GRAM NEGATIVE BACTERIA AND THEIR USES THE TRUSTEES OF PRINCETON UNIVERSITY (US) 2015-03-26 WO disclosed
CN-101426786-A Benzazole potentiators of metabotropic glutamate receptors MERCK & CO INC (US) 2009-05-06 CN disclosed