SCHEMBL16598348

SCHEMBL16598348

NC(N)=NCC(=O)Nc1ccc(C[C@@H](C(=O)O)N(C(=O)[C@@H]2CCCN2)S(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 13/20 0.39
ITGAV P06756 10/20 0.39
ITGA5 P08648 4/20 0.38
CTSC P53634 2/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
ITGB5 P18084 1/20 0.36
TERT O14746 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3113683 0.83 CTSC (0.47) CTSCKMT2A
SCHEMBL3113689 0.83 CTSC (0.47) CTSCKMT2A
SCHEMBL16598553 0.82 ROCK2 (0.37) ITGB1ITGAVITGA5CTSCITGB3
SCHEMBL16598457 0.82 ITGB1 (0.35) ITGB1ITGAVITGA5CTSCITGB3
SCHEMBL19412232 0.77 CTSC (0.39) CTSCMEN1KMT2A
SCHEMBL19412130 0.75 CTSC (0.37) ITGB1ITGA5CTSCITGB3ITGA2B
SCHEMBL27565204 0.74 CTSC (0.47) CTSC
SCHEMBL19412214 0.73 CTSC (0.37) CTSCITGB3ITGA2BTERT
SCHEMBL7450270 0.73 BCHE (0.47) CTSCSMN1; SMN2
SCHEMBL6429094 0.73 CTSC (0.37) CTSCKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3052515-A1 ANTI-ALPHAVBETA1 INTEGRIN COMPOUNDS AND METHODS The Regents of the University of California (US) 2016-08-10 EP disclosed
WO-2015048819-A1 ANTI-ALPHAVBETA1 INTEGRIN COMPOUNDS AND METHODS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-04-02 WO disclosed