SCHEMBL6429094

SCHEMBL6429094

O=C(O)[C@H](Cc1cccc2c1C2)N(C(=O)[C@@H]1CCCN1)S(=O)(=O)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSC P53634 2/20 0.37
SCN4A P35499 1/20 0.36
KMT2A Q03164 1/20 0.32
HTR6 P50406 4/20 0.32
KEAP1 Q14145 3/20 0.32
NFE2L2 Q16236 1/20 0.32
ADAMTS5 Q9UNA0 2/20 0.31
CAMK2A Q9UQM7 2/20 0.31
CAMK2G Q13555 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3113683 0.86 CTSC (0.47) CTSCSCN4AKMT2AADAMTS5
SCHEMBL3113689 0.86 CTSC (0.47) CTSCSCN4AKMT2AADAMTS5
SCHEMBL19412232 0.81 CTSC (0.39) CTSCSCN4AKMT2AHTR6ADAMTS5
SCHEMBL27565204 0.76 CTSC (0.47) CTSCSCN4AADAMTS5
SCHEMBL19412130 0.76 CTSC (0.37) CTSCSCN4AKMT2A
SCHEMBL19412214 0.76 CTSC (0.37) CTSCSCN4AHTR6
SCHEMBL7069746 0.74 ADAMTS5 (0.46) KMT2AKEAP1NFE2L2ADAMTS5
SCHEMBL16598348 0.73 ITGB1 (0.39) CTSCKMT2A
SCHEMBL19412253 0.72 CTSC (0.34) CTSCSCN4A
SCHEMBL19412225 0.71 PRCP (0.34) CTSCSCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP disclosed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP disclosed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO disclosed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed