SCHEMBL1660949

SCHEMBL1660949

O=[C]c1ccccc1C(=O)CCc1ccc(O)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.69
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
SLC5A1 P13866 3/20 0.49
SLC5A2 P31639 3/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
ESR1 P03372 2/20 0.49
KDM4E B2RXH2 1/20 0.49
SLC16A3 O15427 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
TTR P02766 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
POLB P06746 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
THRB P10828 1/20 0.49
SLC2A1 P11166 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11397439 0.88 KEAP1 (0.52) CYP19A1SLC5A1SLC5A2GAAMAPT
SCHEMBL14141727 0.82 CYP19A1 (0.42) CYP19A1MEN1KMT2AGAAMAPT
SCHEMBL1841587 0.81 CYP19A1 (1.00) CYP19A1MEN1KMT2ASLC5A1SLC5A2
SCHEMBL8800760 0.78 CYP19A1 (0.39) CYP19A1MEN1KMT2AGAAMAPT
SCHEMBL210134 0.76 HPGD (0.44) CYP19A1MEN1KMT2AMAPTKDM4E
SCHEMBL1076586 0.74 DPP4 (0.67) CYP19A1MEN1KMT2ASLC5A1SLC5A2
SCHEMBL10936614 0.73 KDM6B (0.51) CYP19A1KDM4ELMNACYP1A2CYP3A4
SCHEMBL4164418 0.73 CYP19A1 (0.61) CYP19A1MEN1KMT2ASLC5A1SLC5A2
SCHEMBL7044239 0.73 LIG1 (0.61) CYP19A1MEN1KMT2AGAAMAPT
SCHEMBL936740 0.72 HTT (0.47) MEN1KMT2AMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2491051-A2 GADD45BETA TARGETING AGENTS Imperial Innovations Limited (GB) 2012-08-29 EP claimed
WO-2011048390-A2 GADD45BETA TARGETING AGENTS IMPERIAL INNOVATIONS LIMITED (GB) 2011-04-28 WO claimed
US-4686283-A POLYPEPTIDES SYNTEX (U.S.A.) INC. (US) 1987-08-11 US disclosed