SCHEMBL10936614

SCHEMBL10936614

O=[C]c1cnccc1C(=O)CCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM6B O15054 7/20 0.51
KDM4C Q9H3R0 7/20 0.51
KDM4D Q6B0I6 4/20 0.51
EGLN3 Q9H6Z9 1/20 0.51
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
LMNA P02545 1/20 0.44
FFAR1 O14842 1/20 0.44
TBXAS1 P24557 2/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1B1 Q16678 1/20 0.43
KDM4E B2RXH2 1/20 0.43
KDM4A O75164 1/20 0.43
KEAP1 Q14145 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
FAAH O00519 1/20 0.40
CYP19A1 P11511 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11397439 0.83 KEAP1 (0.52) FFAR1CYP1A1CYP1B1KEAP1TDP1
SCHEMBL7194181 0.75 KDM4C (0.41) KDM6BKDM4CKDM4DCYP1A2CYP3A4
SCHEMBL4581478 0.74 KMT2A (0.52) KDM6BKDM4CKDM4DCYP1A2CYP3A4
SCHEMBL1660949 0.73 CYP19A1 (0.69) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL11304333 0.72 TDP1 (0.62) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL3247901 0.71 PLOD2 (0.65) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL30965433 0.71 PLOD2 (0.65) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL14141727 0.70 CYP19A1 (0.42) CYP1A2CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL5610674 0.70 TDP1 (0.52) KDM6BKDM4CKDM4DKDM4EKDM4A
SCHEMBL5610323 0.70 KDM4C (0.41) KDM6BKDM4CKDM4DCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148883-A1 ALLOPURINOL PRODRUGS. GEA AS (DK) 1985-07-24 EP disclosed
WO-1985000368-A1 ALLOPURINOL PRODRUGS A/S GEA (DK) 1985-01-31 WO disclosed