SCHEMBL16610073

SCHEMBL16610073

CC(=O)Oc1ccc(C)cc1C(=O)Oc1ccc(CO[Si](C)(C)C(C)(C)C)cc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.44
KMT2A Q03164 3/20 0.42
CFD P00746 1/20 0.39
LMNA P02545 1/20 0.38
HSD17B10 Q99714 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610070 0.91 PTGS2 (0.44) PTGS2KMT2ALMNAHSD17B10KDM4E
SCHEMBL16610075 0.88 PTGS2 (0.46) PTGS2KMT2ACFDLMNAHSD17B10
SCHEMBL22502970 0.87 PTGS2 (0.56) PTGS2KMT2ACFDLMNAHSD17B10
SCHEMBL16610055 0.85 PTGS2 (0.61) PTGS2KMT2ALMNAHSD17B10KDM4E
SCHEMBL18020583 0.84 MAPT (0.42) KMT2AMAPTALDH1A1ATML3MBTL1
SCHEMBL18020601 0.81 PTGS2 (0.53) PTGS2KMT2ACFDLMNAHSD17B10
SCHEMBL12909500 0.81 LMNA (0.44) KMT2ALMNAHSD17B10POLBMAPT
SCHEMBL16599395 0.80 PTGS2 (0.55) PTGS2KMT2ACFDLMNAHSD17B10
SCHEMBL22502975 0.80 MAPT (0.54) PTGS2KMT2AHSD17B10KDM4EMAPT
SCHEMBL16610064 0.79 PTGS2 (0.51) PTGS2KMT2ACFDLMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3049386-B9 COMPOUNDS USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES UNIV KOELN (DE) 2020-11-18 EP disclosed
US-10793509-B2 Compounds useful in the treatment of neoplastic diseases UNIVERSITÄT ZU KOLN (DE) 2020-10-06 US disclosed
EP-3049386-B1 COMPOUNDS USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES UNIV KOELN (DE) 2020-07-22 EP disclosed
US-20160237023-A1 COMPOUNDS USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES UNIVERSITÄT ZU KÖLN (DE) 2016-08-18 US disclosed
US-20160237023-A1 COMPOUNDS USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES UNIVERSITÄT ZU KÖLN (DE) 2016-08-18 US disclosed
WO-2015044177-A1 COMPOUNDS USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES UNIVERSITÄT ZU KÖLN (DE) 2015-04-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160237023-A1 COMPOUNDS USEFUL IN THE TREATMENT OF NEOPLASTIC DISEASES APC, BRCA1, VHL PTGS2 514/4885KMT2A 3041/4885CFD 3054/4885
US-10793509-B2 Compounds useful in the treatment of neoplastic diseases APC, BRCA1, VHL PTGS2 514/4885KMT2A 3041/4885CFD 3054/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.