SCHEMBL16610342

SCHEMBL16610342

CC(C)CNC(=O)/C=C/c1cc([N+](=O)[O-])c([N+](=O)[O-])c(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.42
SMN1; SMN2 Q16637 4/20 0.41
ALDH1A1 P00352 4/20 0.41
AR P10275 4/20 0.41
LMNA P02545 2/20 0.41
CYP3A4 P08684 2/20 0.41
CES2 O00748 1/20 0.41
ABCB11 O95342 1/20 0.41
CYP1A2 P05177 1/20 0.41
GLA P06280 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CHRM1 P11229 1/20 0.41
CYP2C9 P11712 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
TBXA2R P21731 1/20 0.41
AADAC P22760 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP2C19 P33261 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610337 0.78 TRPV1 (0.46) TRPV1SMN1; SMN2ALDH1A1LMNACYP3A4
SCHEMBL28013192 0.78 ALDH1A1 (0.45) SMN1; SMN2ALDH1A1HTTBACE1HPGD
SCHEMBL16610336 0.77 TRPV1 (0.52) TRPV1SMN1; SMN2ALDH1A1CYP3A4CYP1A2
SCHEMBL28012614 0.77 TRPV1 (0.52) TRPV1SMN1; SMN2ALDH1A1CYP3A4CYP1A2
SCHEMBL16610366 0.76 TRPV1 (0.46) TRPV1SMN1; SMN2ALDH1A1CYP3A4CYP1A2
SCHEMBL16610453 0.75 AR (0.37) SMN1; SMN2ALDH1A1ARLMNACYP3A4
SCHEMBL28013193 0.75 TRPV1 (0.51) TRPV1SMN1; SMN2LMNAHTTBACE1
SCHEMBL16610380 0.75 TRPV1 (0.51) TRPV1SMN1; SMN2LMNAHTTBACE1
SCHEMBL16610410 0.73 TRPV1 (0.57) TRPV1SMN1; SMN2ALDH1A1CYP3A4CYP1A2
SCHEMBL16610369 0.73 TRPV1 (0.60) TRPV1ALDH1A1LMNACYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed