SCHEMBL16610375

SCHEMBL16610375

COc1cc(/C=C/C(=O)N2CCCCC2)cc(C(F)(F)F)c1OC

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.75
KDM4E B2RXH2 6/20 0.75
HPGD P15428 3/20 0.75
KMT2A Q03164 2/20 0.59
TRPV1 Q8NER1 1/20 0.59
TP53 P04637 3/20 0.54
MAPT P10636 2/20 0.54
HSD17B10 Q99714 2/20 0.54
STAT6 P42226 1/20 0.54
MEN1 O00255 1/20 0.53
ATM Q13315 1/20 0.53
BCHE P06276 3/20 0.53
MAOA P21397 3/20 0.53
ACHE P22303 3/20 0.53
MAOB P27338 3/20 0.53
APP P05067 2/20 0.50
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C19 P33261 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610371 0.88 ALDH1A1 (0.60) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL27183471 0.88 ALDH1A1 (0.97) ALDH1A1KDM4EHPGDKMT2ATRPV1
Cinoctramide SCHEMBL2111109 0.88 ALDH1A1 (0.97) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL15884182 0.81 ALDH1A1 (0.78) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL16610368 0.80 KDM4E (0.72) ALDH1A1KDM4EHPGDHSD17B10ATM
SCHEMBL19187350 0.80 ALDH1A1 (0.76) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL25309070 0.79 ALDH1A1 (0.80) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL11717607 0.79 ALDH1A1 (0.79) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL11753535 0.78 ALDH1A1 (0.81) ALDH1A1KDM4EHPGDKMT2ATRPV1
SCHEMBL16610374 0.77 ALOX5 (0.61) ALDH1A1KDM4EHPGDKMT2ATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed