SCHEMBL16610412

SCHEMBL16610412

O=C(O)/C=C/c1cc(OC(F)F)c(OC(F)F)c(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.46
ALDH1A1 P00352 5/20 0.46
HPGD P15428 3/20 0.46
HSD17B10 Q99714 2/20 0.46
HTR1A P08908 1/20 0.46
HTR2C P28335 1/20 0.46
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
PKM P14618 2/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GAA P10253 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
APP P05067 2/20 0.38
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610391 0.80 TRPV1 (0.49) KDM4EALDH1A1HPGDHTR1AHTR2C
SCHEMBL28012610 0.80 TRPV1 (0.49) KDM4EALDH1A1HPGDHTR1AHTR2C
SCHEMBL16610418 0.80 DRD1 (0.39)
SCHEMBL16610368 0.78 KDM4E (0.72) KDM4EALDH1A1HPGDHSD17B10HTR1A
SCHEMBL16610425 0.78 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10HTR1A
SCHEMBL16048499 0.77 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10HTR1A
SCHEMBL16048498 0.77 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10HTR1A
SCHEMBL142116 0.74 KDM4E (0.59) KDM4EALDH1A1HPGDHSD17B10HTR1A
SCHEMBL16610372 0.72 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10HTR1A
SCHEMBL16610417 0.72 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed