SCHEMBL16610417

SCHEMBL16610417

CCCCOc1cc(/C=C/C(=O)O)cc(C(F)(F)F)c1OCCCC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.48
AKR1C3 P42330 2/20 0.47
POLB P06746 1/20 0.46
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
HTR1A P08908 3/20 0.45
HTR2C P28335 3/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
GAA P10253 2/20 0.44
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
ACHE P22303 3/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
APP P05067 1/20 0.40
RXRA P19793 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16610334 0.88 THRB (0.44) KDM4EAKR1C3POLBKMT2AMEN1
SCHEMBL16610426 0.87 THRA (0.40) KDM4EAKR1C3POLBKMT2AMEN1
SCHEMBL16610416 0.87 HTR1A (0.43) KDM4EAKR1C3POLBKMT2AMEN1
SCHEMBL16610411 0.86 APP (0.41) KMT2AMEN1HTR1AHTR2CALDH1A1
SCHEMBL16610407 0.82 ALDH1A1 (0.39) KDM4EPOLBKMT2AMEN1ALDH1A1
SCHEMBL6023949 0.79 PKM (0.62) KDM4EAKR1C3POLBKMT2AMEN1
SCHEMBL6023916 0.79 PKM (0.62) KDM4EAKR1C3POLBKMT2AMEN1
SCHEMBL16610368 0.77 KDM4E (0.72) KDM4EHTR1AHTR2CALDH1A1HPGD
SCHEMBL16610422 0.76 THRB (0.46) KDM4EAKR1C3POLBKMT2AMEN1
SCHEMBL16048499 0.76 KDM4E (0.61) KDM4EPOLBHTR1AHTR2CALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed