SCHEMBL16610372

SCHEMBL16610372

COc1c(O)cc(/C=C/C(=O)O)cc1C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.55
ALDH1A1 P00352 5/20 0.55
HSD17B10 Q99714 4/20 0.55
HPGD P15428 4/20 0.55
HTR1A P08908 1/20 0.55
HTR2C P28335 1/20 0.55
PKM P14618 2/20 0.51
PTGS1 P23219 1/20 0.51
PTGS2 P35354 1/20 0.51
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA3 P07451 2/20 0.48
CA4 P22748 2/20 0.48
CA6 P23280 2/20 0.48
CA5A P35218 2/20 0.48
CA7 P43166 2/20 0.48
CA9 Q16790 2/20 0.48
CA14 Q9ULX7 2/20 0.48
CA5B Q9Y2D0 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16048498 0.91 KDM4E (0.61) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL16048499 0.91 KDM4E (0.61) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL16610368 0.86 KDM4E (0.72) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL16610422 0.85 THRB (0.46) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL20600978 0.85 KDM4E (0.69) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL21852876 0.85 KDM4E (0.69) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL16610334 0.82 THRB (0.44) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL16610370 0.80 ALDH1A1 (0.45) KDM4EALDH1A1HPGDPTGS2CA1
SCHEMBL16610371 0.80 ALDH1A1 (0.60) KDM4EALDH1A1HSD17B10HPGDAPP
SCHEMBL16610410 0.79 TRPV1 (0.57) KDM4EALDH1A1HTR1AHTR2CPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015043522-A1 TRIFLUOROMETHYL-CONTAINING AMIDE ALKALOID, MANUFACTURING METHOD AND PHARMACEUTICAL USE THEREOF 天士力制药集团股份有限公司 2015-04-02 WO disclosed