SCHEMBL16612059

SCHEMBL16612059

COc1cc(C)c(CS)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
IDO1 P14902 1/20 0.43
CYP3A4 P08684 3/20 0.39
HPGD P15428 3/20 0.38
TAAR1 Q96RJ0 1/20 0.38
MEN1 O00255 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
FFAR4 Q5NUL3 1/20 0.35
PTPN1 P18031 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ACHE P22303 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14363077 0.87 ALDH1A1 (0.39) ALDH1A1IDO1CYP3A4HPGDTAAR1
SCHEMBL14963168 0.87 ALDH1A1 (0.41) ALDH1A1IDO1CYP3A4HPGDPTPN1
SCHEMBL13067432 0.78 ALDH1A1 (0.48) ALDH1A1CYP3A4HPGDTAAR1MEN1
SCHEMBL5730733 0.76 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDTAAR1MEN1
SCHEMBL10753734 0.76 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDTAAR1MEN1
SCHEMBL15216746 0.76 ALDH1A1 (0.46) ALDH1A1CYP3A4HPGDTAAR1MEN1
SCHEMBL2332266 0.76 ALDH1A1 (0.46) ALDH1A1IDO1CYP3A4CYP1A1CYP1B1
SCHEMBL9171915 0.74 ALDH1A1 (0.43) ALDH1A1IDO1CYP3A4TAAR1CYP1A1
SCHEMBL509722 0.74 HRH3 (0.40) ALDH1A1IDO1MEN1TSHRKMT2A
SCHEMBL21938394 0.73 NOS3 (0.43) ALDH1A1CYP3A4HPGDTAAR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2857388-A1 Azoles containing sulfone Grünenthal GmbH (DE) 2015-04-08 EP disclosed