SCHEMBL16612830

SCHEMBL16612830

Nc1cnn(CCOc2cccc(F)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HCRTR2 O43614 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
MAPT P10636 2/20 0.43
LMNA P02545 1/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GRM5 P41594 4/20 0.42
HDAC6 Q9UBN7 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALK Q9UM73 1/20 0.39
DCPS Q96C86 1/20 0.38
JAK2 O60674 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12479353 0.84 MEN1 (0.64) MEN1KMT2AHCRTR2MAPTLMNA
SCHEMBL16612776 0.83 MAPT (0.55) MEN1KMT2AHCRTR2HDAC1HDAC2
SCHEMBL16612864 0.83 MEN1 (0.47) MEN1KMT2AHDAC1HDAC2MAPT
SCHEMBL12479925 0.76 MAPT (0.50) MEN1KMT2AHCRTR2MAPTLMNA
SCHEMBL16613012 0.75 MAPT (0.49) MEN1KMT2AHCRTR2HDAC1HDAC2
SCHEMBL12479530 0.73 MAOB (0.50) MEN1KMT2AHCRTR2MAPTALDH1A1
SCHEMBL3616273 0.73 MAPT (0.65) MEN1KMT2AMAPTLMNAALDH1A1
Hydrochloric Acid SCHEMBL21523747 0.71 MAPT (0.68) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL16612785 0.70 HCRTR2 (0.46) MEN1KMT2AHCRTR2MAPTLMNA
Fluorobenzene SCHEMBL27885840 0.70 MAPT (0.53) MEN1KMT2AMAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP disclosed