SCHEMBL16612941

SCHEMBL16612941

O=C(O)Oc1ncoc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.46
IP6K3 Q96PC2 1/20 0.46
IP6K2 Q9UHH9 1/20 0.46
KMO O15229 2/20 0.45
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
NOTUM Q6P988 2/20 0.44
ALDH1A1 P00352 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.40
XDH P47989 1/20 0.40
KDM4E B2RXH2 1/20 0.40
PIN1 Q13526 1/20 0.40
CNR2 P34972 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
PARP1 P09874 1/20 0.39
SCN2A Q99250 1/20 0.39
KIF11 P52732 1/20 0.39
CTSK P43235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612942 0.84 GSK3B (0.47) KIF11
SCHEMBL16612795 0.83 KDM4E (0.43) KMONOTUMALDH1A1SMN1; SMN2KDM4E
SCHEMBL16612958 0.82 STK17B (0.43) ALDH1A1XDHKDM4ECYP1A2
SCHEMBL16612946 0.82 ADORA2A (0.44) IP6K1IP6K3IP6K2KMOALDH1A1
SCHEMBL5546097 0.80 ADORA2A (0.54) ALDH1A1KDM4ECYP1A2
SCHEMBL1167600 0.80 KMO (0.51) IP6K1IP6K3IP6K2KMORXRA
SCHEMBL16613030 0.80 KMO (0.42) KMORXRARXRBRXRGNOTUM
SCHEMBL15189624 0.80 MEN1 (0.46) IP6K1IP6K3IP6K2KMORXRA
SCHEMBL15189706 0.78 GSK3B (0.51) RXRARXRBNOTUMALDH1A1SMN1; SMN2
SCHEMBL16612913 0.78 NOTUM (0.45) NOTUMXDHPIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed