SCHEMBL16612913

SCHEMBL16612913

N#Cc1cccc(-c2ocnc2OC(=O)O)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
CLK4 Q9HAZ1 1/20 0.43
XDH P47989 1/20 0.43
SLC22A12 Q96S37 1/20 0.43
PTGDR2 Q9Y5Y4 2/20 0.41
F11 P03951 1/20 0.41
PIN1 Q13526 1/20 0.41
HCRTR2 O43614 1/20 0.40
EGLN1 Q9GZT9 2/20 0.39
FAAH O00519 1/20 0.39
GRK6 P43250 1/20 0.38
PRKDC P78527 1/20 0.38
ATR Q13535 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
ADORA2A P29274 1/20 0.38
HPGDS O60760 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRG2 P18507 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16612946 0.83 ADORA2A (0.44) ADORA2A
SCHEMBL5546097 0.81 ADORA2A (0.54) HCRTR2ADORA2A
SCHEMBL16612795 0.81 KDM4E (0.43) NOTUMPIN1HCRTR2EGLN1ADORA2A
SCHEMBL1167684 0.81 PIN1 (0.51) NOTUMCLK4XDHSLC22A12PTGDR2
SCHEMBL15189624 0.81 MEN1 (0.46) HCRTR2ADORA2A
SCHEMBL16613030 0.81 KMO (0.42) NOTUMHCRTR2ADORA2A
SCHEMBL15189706 0.79 GSK3B (0.51) NOTUMCLK4PIN1
SCHEMBL16612964 0.78 NOTUM (0.44) NOTUMHCRTR2ADORA2A
SCHEMBL16612941 0.78 IP6K1 (0.46) NOTUMXDHPIN1
SCHEMBL6286017 0.78 NOTUM (0.44) NOTUMCLK4XDHSLC22A12PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2675801-B1 NOVEL PYRAZOLE AND IMIDAZOLE DERIVATIVES USEFUL AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2015-04-08 EP claimed