SCHEMBL16615221

SCHEMBL16615221

O=C(NCCc1ccccc1)c1c2c3c(n1-2)NCCN3Cc1c(Cl)ccc(F)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
MAPT P10636 3/20 0.39
TP53 P04637 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.36
PTGS2 P35354 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MCHR1 Q99705 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615202 0.77 MAPT (0.42) MAPTTP53SMN1; SMN2ALDH1A1LMNA
SCHEMBL20859464 0.69 MAPT (0.41) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL17969745 0.67 KDM4E (0.39) MAPTALDH1A1KDM4E
SCHEMBL20859307 0.66 PLAAT3 (0.33) L3MBTL1MAPTTP53SMN1; SMN2NPC1
SCHEMBL17969728 0.65 ALK (0.49)
SCHEMBL16615279 0.64 HDAC1 (0.33)
SCHEMBL16615259 0.63 GAA (0.41) MAPTTP53SMN1; SMN2NPC1RAB9A
SCHEMBL16615167 0.62 MAP4K3 (0.31)
SCHEMBL14456882 0.58 MCHR1 (0.60) SMN1; SMN2NPC1RAB9AALDH1A1KDM4E
SCHEMBL16615321 0.58 ALK (0.48) MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050884-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES Limited Liability Company "National Pharmaceutical (RU) 2016-08-03 EP disclosed
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed