SCHEMBL16615282

SCHEMBL16615282

O=C(Nc1ccc(N2CCOCC2)cc1)c1cc2c(nn1)NCCN2Cc1c(Cl)ccc(F)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.44
RAB9A P51151 5/20 0.42
NPC1 O15118 4/20 0.42
MAPT P10636 7/20 0.41
LMNA P02545 3/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
PDE7A Q13946 3/20 0.41
RAF1 P04049 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
ALDH1A1 P00352 2/20 0.40
MITF O75030 1/20 0.40
TP53 P04637 1/20 0.40
CFTR P13569 1/20 0.40
HPGD P15428 1/20 0.40
DGAT1 O75907 1/20 0.39
TSHR P16473 1/20 0.39
PRKAA2 P54646 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17918849 0.90 MET (0.43) NPC1MAPTLMNAHTTMEN1
SCHEMBL17918706 0.86 MAPT (0.44) RAB9ANPC1MAPTLMNAHTT
SCHEMBL17918718 0.85 CFTR (0.42) NPC1MAPTLMNAHTTMEN1
SCHEMBL17918788 0.85 RAB9A (0.46) NTRK1RAB9ANPC1MAPTLMNA
SCHEMBL16615212 0.84 MET (0.45) RAB9ANPC1MAPTMEN1KMT2A
SCHEMBL17918716 0.82 ALK (0.46) MAPTLMNASMN1; SMN2ALDH1A1HPGD
SCHEMBL18106085 0.82 MET (0.54) NTRK1MEN1KMT2ACFTR
SCHEMBL16615218 0.81 SETD2 (0.37) NTRK1MAPTALDH1A1
SCHEMBL17918705 0.81 NTRK1 (0.54) NTRK1RAB9ANPC1MAPTLMNA
SCHEMBL17969779 0.81 NTRK1 (0.50) NTRK1RAB9ANPC1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed