SCHEMBL16615218

SCHEMBL16615218

CNC1CCN(c2cccc(NC(=O)c3cc4c(nn3)NCCN4Cc3c(Cl)ccc(F)c3Cl)c2)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SETD2 Q9BYW2 5/20 0.37
NSD2 O96028 1/20 0.37
ALK Q9UM73 2/20 0.37
IDO1 P14902 1/20 0.37
PLK4 O00444 1/20 0.37
JAK2 O60674 1/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
ABL1 P00519 1/20 0.37
LCK P06239 1/20 0.37
CSF1R P07333 1/20 0.37
RET P07949 1/20 0.37
MET P08581 1/20 0.37
ROS1 P08922 1/20 0.37
FGFR1 P11362 1/20 0.37
SRC P12931 1/20 0.37
FER P16591 1/20 0.37
FGFR3 P22607 1/20 0.37
LTK P29376 1/20 0.37
FLT4 P35916 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17918850 0.91 SETD2 (0.48) SETD2NSD2ALKIDO1PLK4
SCHEMBL16615283 0.82 SETD2 (0.38) SETD2NSD2IDO1ALDH1A1MALT1
SCHEMBL16615282 0.81 NTRK1 (0.44) ALDH1A1MAPTNTRK1
SCHEMBL17918788 0.79 RAB9A (0.46) ALDH1A1MAPTCYP3A4NTRK1
SCHEMBL17918715 0.78 KCNQ2 (0.44) ALKALDH1A1MAPTKDM4E
SCHEMBL18106050 0.78 ALK (0.51) SETD2ALKJAK2PRKD3MAP4K4
SCHEMBL16615153 0.77 PLK4 (0.41) ALKPLK4JAK2PRKD3MAP4K4
SCHEMBL17969758 0.77 EGFR (0.39) ALKPLK4JAK2PRKD3MAP4K4
SCHEMBL16615212 0.77 MET (0.45) ALKPLK4JAK2PRKD3MAP4K4
SCHEMBL18106085 0.77 MET (0.54) ALKPLK4JAK2PRKD3MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed