SCHEMBL16615322

SCHEMBL16615322

ClC1=CC2=C(NCCN2Cc2cc(Cl)ccc2Cl)NN1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.42
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.38
P2RX7 Q99572 1/20 0.37
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
DBH P09172 1/20 0.36
MAOB P27338 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
GPR6 P46095 5/20 0.33
CYP2A13 Q16696 1/20 0.33
PKM P14618 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
HTR1A P08908 1/20 0.32
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32
PIK3CA P42336 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17969806 0.78 BCHE (0.35) ALKDRD2DRD3KCNH2P2RX7
SCHEMBL17969755 0.76 ALK (0.34) ALKGPR6
SCHEMBL16615210 0.74 THRB (0.36) ALKDRD2DRD3KCNH2MAPT
SCHEMBL17969746 0.73 MAPT (0.43) MAPT
SCHEMBL20859430 0.71 PLK4 (0.35) ALK
SCHEMBL20859370 0.68 DRD2 (0.39) ALKDRD2DRD3KCNH2P2RX7
SCHEMBL20859362 0.68 ALK (0.34) ALKDRD2DRD3KCNH2P2RX7
SCHEMBL3960485 0.68 SLC6A2 (0.52) DRD2DRD3KCNH2DBHSLC6A2
SCHEMBL14387479 0.68 ALK (0.61) ALKDRD2DRD3KCNH2P2RX7
SCHEMBL17918668 0.68 ALK (0.53) ALKDRD2DRD3KCNH2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed