SCHEMBL16615210

SCHEMBL16615210

Clc1ccc(Cl)c(CN2CCNC3=C2C=C(c2nnc(C4CCNCC4)o2)NN3)c1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.36
ALK Q9UM73 1/20 0.34
KCNH2 Q12809 2/20 0.33
LRRK2 Q5S007 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
MAPT P10636 2/20 0.33
ALOX15B O15296 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GPR6 P46095 5/20 0.32
TP53 P04637 2/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
OPRM1 P35372 1/20 0.32
GPR4 P46093 1/20 0.32
HTR3A P46098 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20859343 0.84 ALK (0.36) THRBALKKCNH2LRRK2DRD2
SCHEMBL20859264 0.78 PLK4 (0.34) ALKKCNH2LRRK2DRD2DRD3
SCHEMBL16615325 0.78 ALK (0.44) THRBALKKCNH2LRRK2DRD2
SCHEMBL16615323 0.78 ALK (0.40) THRBALKKCNH2LRRK2DRD2
SCHEMBL17969755 0.75 ALK (0.34) ALKLRRK2GPR6
SCHEMBL16615322 0.74 ALK (0.42) ALKKCNH2DRD2DRD3MAPT
SCHEMBL17969806 0.73 BCHE (0.35) ALKKCNH2DRD2DRD3GPR6
SCHEMBL16615324 0.73 ALK (0.34) THRBALKKCNH2DRD2DRD3
SCHEMBL20859351 0.72 THRB (0.35) THRBALK
SCHEMBL20859451 0.71 ENPP2 (0.33) THRBALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050884-B1 NEW CHEMICAL COMPOUNDS (DERIVATIVES) AND THEIR APPLICATION FOR THE TREATMENT OF ONCOLOGICAL DISEASES LIMITED LIABILITY COMPANY NATIONAL PHARMACEUTICAL TECH (RU) 2019-04-03 EP disclosed
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed