SCHEMBL16615323

SCHEMBL16615323

Clc1ccc(Cl)c(CN2CCNc3[nH]c(-c4nnc(C5CCNCC5)o4)cc32)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.40
THRB P10828 1/20 0.37
PLAT P00750 5/20 0.33
LRRK2 Q5S007 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
KCNH2 Q12809 1/20 0.33
ALOX15B O15296 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615325 0.82 ALK (0.44) ALKTHRBLRRK2DRD2DRD3
SCHEMBL16615361 0.78 ALK (0.41) ALKLRRK2DRD2DRD3KCNH2
SCHEMBL16615210 0.78 THRB (0.36) ALKTHRBLRRK2DRD2DRD3
SCHEMBL20859343 0.76 ALK (0.36) ALKTHRBPLATLRRK2DRD2
SCHEMBL16615084 0.75 ALK (0.46) ALKLRRK2DRD2DRD3KCNH2
SCHEMBL16615287 0.75 ALK (0.44) ALKLRRK2DRD2DRD3KCNH2
SCHEMBL16615290 0.75 ALK (0.38) ALKTP53
SCHEMBL17918694 0.75 ALK (0.49) ALKLRRK2DRD2DRD3KCNH2
SCHEMBL16615324 0.74 ALK (0.34) ALKTHRBDRD2DRD3KCNH2
SCHEMBL17918756 0.72 TLR9 (0.39) ALKTHRBLRRK2TP53SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3050884-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES Limited Liability Company "National Pharmaceutical (RU) 2016-08-03 EP disclosed
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed