SCHEMBL16615324

SCHEMBL16615324

Clc1ccc(Cl)c(CN2CCNc3c2c2c(-c4nnc(C5CCNC5)o4)n3-2)c1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.34
THRB P10828 1/20 0.33
TLR9 Q9NR96 2/20 0.32
TLR8 Q9NR97 2/20 0.32
TLR7 Q9NYK1 2/20 0.32
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
KCNH2 Q12809 1/20 0.31
TP53 P04637 1/20 0.30
ALOX15B O15296 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TNKS O95271 1/20 0.30
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16615327 0.89 ALK (0.40) ALKDRD2DRD3KCNH2TP53
SCHEMBL16615266 0.85 LMNA (0.38) ALKTLR9TLR8TLR7ALDH1A1
SCHEMBL16615328 0.79 ALK (0.43) ALKDRD2DRD3KCNH2TP53
SCHEMBL16615186 0.78 ALK (0.34) ALK
SCHEMBL16615265 0.75 NPC1 (0.43) ALKKCNH2ALDH1A1
SCHEMBL16615325 0.74 ALK (0.44) ALKTHRBDRD2DRD3KCNH2
SCHEMBL16615323 0.74 ALK (0.40) ALKTHRBDRD2DRD3KCNH2
SCHEMBL16615365 0.74 PLK4 (0.35) ALKDRD2DRD3KCNH2TP53
SCHEMBL16615210 0.73 THRB (0.36) ALKTHRBDRD2DRD3KCNH2
SCHEMBL16615276 0.72 ALK (0.32) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015047133-A1 NOVEL CHEMICAL COMPOUNDS (VARIANTS) AND THE USE THEREOF TO TREAT ONCOLOGICAL DISEASES ОБЩЕСТВО С ОГРАНИЧЕННОЙ ОТВЕТСТВЕННОСТЬЮ "ОТЕЧЕСТВЕННЫЕ ФАРМАЦЕВТИЧЕСКИЕ ТЕХНОЛОГИИ" 2015-04-02 WO disclosed