SCHEMBL16622143

SCHEMBL16622143

CCc1nc(N)nc(N)c1OCCO

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 14/20 0.58
HEXA P06865 3/20 0.42
HEXB P07686 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12487673 0.90 DHFR (0.59) DHFRHEXAHEXB
SCHEMBL16622144 0.80 DHFR (0.63) DHFRHEXAHEXB
SCHEMBL18670791 0.75 DHFR (0.47) DHFRHEXAHEXB
SCHEMBL12487396 0.74 DHFR (1.00) DHFRHEXAHEXB
Hydrochloric Acid SCHEMBL12486624 0.73 DHFR (1.00) DHFRHEXAHEXB
Hydrochloric Acid SCHEMBL11183905 0.72 DHFR (0.78) DHFRHEXAHEXB
SCHEMBL31155811 0.72 DHFR (0.91) DHFR
SCHEMBL31155818 0.71 DHFR (0.41) DHFRHEXAHEXB
SCHEMBL12487404 0.71 DHFR (1.00) DHFRHEXAHEXB
SCHEMBL3267488 0.71 DHFR (0.80) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9000003-B2 Anti-folate antimalarials with dual-binding modes and their preparation NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2015-04-07 US disclosed
US-9000003-B2 Anti-folate antimalarials with dual-binding modes and their preparation NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2015-04-07 US disclosed